Search Result "4-Thiadiazole derivatives"


Synthesis of Some Novel 2-Azetidinones/4-Thiazolidinones Bearing 1, 3, 4- Thiadiazole Nucleus and Screening for its Anti-Imflammatory Activity

Journal: Letters in Drug Design & Discovery
Volume: 13 Issue: 7 Year: 2016 Page: 676-683
Author(s): B. Gowramma, T. K. Praveen, R. Kalirajan, B. Babu

Research Article

Synthesis, Antimicrobial Evaluation of Some New 1, 3, 4-Thiadiazoles and 1, 3, 4- Thiadiazines

Journal: Current Organic Synthesis
Volume: 15 Issue: 8 Year: 2018 Page: 1161-1170
Author(s): Ameen A. Abu-Hashem,Rasha A. M. Faty

Research Article

Design, Synthesis, Molecular Docking and In silico Analysis of Some Novel 2-Amino-1, 3, 4-Thiadiazole Derivatives as Potent DNA Gyrase B Inhibitors

Journal: Current Bioactive Compounds
Volume: 17 Issue: 7 Year: 2021 Page: 8-17
Author(s): Natarajan Ramalakshmi,Prabakaran A.,Sumithra S.,Keerthika S.,Nivetha J.,Raveena R.

Synthesis, Cytotoxic Evaluation, Docking and QSAR Study of N-(4-Oxo- 2-(4-((5-Aryl-1,3,4-Thiadiazol-2-yl)Amino)Phenyl)Thiazolidin-3-yl) Benzamides as Antitubulin Agents

Journal: Current Topics in Medicinal Chemistry
Volume: 16 Issue: 2 Year: 2016 Page: 2509-2520
Author(s): Chawla Amit, Chawla Payal, U.S. Baghel, Deep Aakash

Research Article

Synthesis of Novel 6-(1H-pyrazol-4-yl)-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazoles as Potential Antimicrobial Agents

Journal: Letters in Organic Chemistry
Volume: 15 Issue: 2 Year: 2018 Page: 92-98
Author(s): Rashmi Pundeer,Pooja Ranjan,Richa Prakash,Radhika Joshi

One-Pot Synthesis of 1,3-Thiazolidin-4-Ones Derivatives from 2-Amino-1,3,4-Thiadiazole

Journal: Letters in Organic Chemistry
Volume: 4 Issue: 7 Year: 2007 Page: 505-508
Author(s): Wilson Cunico, Claudia R. B. Gomes, Maria de Lourdes G. Ferreira, Liliane R. Capri, Margareth R. L. Santos, Paula M. Sa, Nubia Boechat, Monica M. Bastos, Lindalva C. Maciel, Lucia M. U. Mayer

Synthesis and Biological Evaluation of Novel N-[(7-pyridin-4-yl-2, 3- dihydro-benzofuran-2-yl) Methyl]-(4-methyl-1, 2, 3-thiadiazole-5-yl) Formamide as a Potent Immunosuppressant Agent

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 3 Year: 2014 Page: 375-379
Author(s): Chen Fan,Yubin Wang,Peng Lu,Xiaojian Xue,Jinxiong She

Research Article

Synthesis and Biological Evaluation of 1,3,4-Thiadiazole Linked Phthalimide Derivatives as Anticancer Agents

Journal: Letters in Drug Design & Discovery
Volume: 14 Issue: 10 Year: 2017 Page: 1138-1144
Author(s): Zahra Rezaei,Setareh Moghimi,Rezvan Javaheri,Mehdi Asadi,Mohammad Mahdavi,Shabnam Shabani,Najmeh Edraki,Omidreza Firuzi,Maliheh Safavi,Mohsen Amini,Ali Asadipour,Elnaz Zeinalzadeh,Loghman Firoozpour,Alireza Foroumadi

Synthesis and Antifungal Activity of 1,2,3-thiadiazole Derivatives Containing 1,3,4-thiadiazole Moiety

Journal: Letters in Drug Design & Discovery
Volume: 11 Issue: 7 Year: 2014 Page: 940-943
Author(s): Shui-Lin Yan, Ming-Yan Yang, Zhao-Hui Sun, Li-Jing Min, Cheng-Xia Tan, Jian-Quan Weng, Hong-Ke Wu, Xing-Hai Liu

Research Article

Synthesis, Antioxidant and Antiurease Activities of Some New 5,6- dichloro-2-(4-fluorobenzyl)-1H-benzimidazole Derivatives Containing Furan, Oxadiazole, Triazole and Thiadiazole Moieties

Journal: Letters in Drug Design & Discovery
Volume: 16 Issue: 8 Year: 2019 Page: 939-947
Author(s): Hakan Bektas,Canan Albay,Emre Menteşe,Bahar Bilgin Sokmen,Zafer Kurt,Dilem Şen

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